Category:
Prophylactic Biological Products
CAS NO:
375815-87-5
Standard:
USP,
Varenicline tartrate is the pharmaceutical salt form of varenicline, a partial agonist at nicotinic acetylcholine receptors. It is synthesized via chiral resolution or asymmetric catalysis to ensure high enantiomeric purity. The compound features the molecular formula C10H14N4O·C4H6O6 and carries CAS No. 159725-28-9.
Strictly contraindicated for patients with severe renal impairment without dose adjustment. Storage requires controlled conditions (20-25°C) in moisture-proof containers. Handling mandates PPE to prevent skin contact and inhalation of dust particles.