Category:
Prophylactic Biological Products
CAS NO:
NA
Standard:
In-house Standards,
Fosaprepitant Dimeglumine is a water-soluble prodrug of aprepitant, serving as a neurokinin-1 (NK1) receptor antagonist. It is synthesized via amide coupling to enhance bioavailability for intravenous administration. Its molecular formula is C24H30ClN4O5 and CAS number is 689837-39-6.
Contraindicated with strong CYP3A4 inducers like rifampin. Store vials at controlled room temperature (20°C to 25°C) protected from light. Avoid mixing with alkaline solutions to prevent hydrolysis of the prodrug structure.