Category:
Prophylactic Biological Products
CAS NO:
NA
Standard:
In-house Standards,
Lopinavir/Ritonavir is a fixed-dose combination of two antiretroviral protease inhibitors used primarily in HIV-1 management. The formulation leverages ritonavir as a pharmacokinetic booster to inhibit CYP3A4, thereby elevating lopinavir plasma concentrations. Molecular Formula: C57H74N10O8; CAS No.: 209686-85-3 (fixed ratio).
Strictly contraindicated with specific CYP3A substrates due to severe interaction risks. Store below 25°C in a dry environment to maintain stability. Monitor hepatic function and lipid profiles during long-term clinical administration.