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Overview
Bilastine is a second-generation antihistamine used for treating allergic rhinitis and urticaria. Produced via organic synthesis, its molecular formula is C21H26N4O2 with CAS No. 197507-87-6.
Application
- Pharmaceutical Manufacturing: Formulation of non-sedating oral tablets for seasonal allergies.
- Clinical Research: Investigational use in chronic spontaneous urticaria protocols.
- Veterinary Medicine: Off-label application for pruritus control in companion animals.
Precautions
Avoid concomitant intake with fruit juices to prevent reduced bioavailability. Store API in a dry, cool environment below 25°C protected from light. Contraindicated in patients with known hypersensitivity or severe renal impairment.